Our recent work on aliphatic CO-to-N atom swap enabled by NAHA chemistry, now online in
@science.org ! Congratulations to Zining, Zhehan and Rong!
www.science.org/doi/10.1126/...
Medicinal chemistry campaigns routinely require access to series of saturated nitrogen heterocycle (SNH)–based analogs that place nitrogen at different positions to probe structure-activity relationsh...