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Delighted to share our publication in @bloodjournal.bsky.social where we describe the identification of antifungal itraconazole as a potent inhibitor of mitochondrial metabolism in AML Great effort by joint first authors Katerina Himonas and Lucie de Beauchamp. ashpublications.org/blood/articl...
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Key Points. Nutrient sensing drug-repurposing screen identifies itraconazole, an FDA-approved azole antifungal, as a mitochondrial metabolism inhibitorItra
ashpublications.org
A metabolism-specific drug-repurposing screen reveals itraconazole as a potent OXPHOS inhibitor in acute myeloid leukemia
Helgason Lab